TEMPO-copper(II) diimine-catalysed oxidation of benzylic alcohols in aqueous media

Pawel J Figiel, Markku Leskelä, Timo Repo

Research output: Contribution to journalArticleScientificpeer-review

Abstract

In situ generated copper(II)-diimine complexes combined with TEMPO (2,2,6,6-tetramethylpiperidinyl-1-oxyl radical) were studied in the oxidation of benzylic alcohols, the focus being on enviromentally benign reaction conditions. In this respect, reactions were studied in aqueous alkaline solutions and dioxygen was used as an end oxidant. This simple catalytic system turned out to be highly efficient and selective in the oxidation of primary and secondary benzylic alcohols to their corresponding carbonyl compounds. Under optimised reaction conditions [5 mol% of TEMPO, 3 mol % of copper(II) diimine, pH 12.6-13.5, 80 degrees C, 1.0 bar O-2] benzyl alcohol was quantitatively and selectively oxidised to benzaldehyde. According to ESI-MS studies, coordination of TEMPO, as well as deprotonated benzyl alcohol to the parent copper-diimine complex in aqueous solutions is feasible. Supported by these observations a plausible reaction mechanism is proposed for the oxidation reaction.
Original languageEnglish
JournalAdvanced Synthesis & Catalysis
Volume349
Issue number7
Pages (from-to)1173-1179
Number of pages7
ISSN1615-4150
DOIs
Publication statusPublished - 2007
MoE publication typeA1 Journal article-refereed

Fields of Science

  • 116 Chemical sciences

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