Recent progress and challenges in screening and characterization of UGT1A1 inhibitors

Xia Lv, Yangliu Xia, Moshe Finel, Jingjing Wu, Guangbo Ge, Ling Yang

Tutkimustuotos: ArtikkelijulkaisuKatsausartikkeliTieteellinenvertaisarvioitu

Alkuperäiskielienglanti
LehtiActa pharmaceutica sinica b
Vuosikerta9
Numero2
Sivut258-278
Sivumäärä21
ISSN2211-3835
DOI - pysyväislinkit
TilaJulkaistu - maaliskuuta 2019
OKM-julkaisutyyppiA2 Katsausartikkeli tieteellisessä aikakauslehdessä

Tieteenalat

  • 116 Kemia
  • 317 Farmasia

Lainaa tätä

Lv, Xia ; Xia, Yangliu ; Finel, Moshe ; Wu, Jingjing ; Ge, Guangbo ; Yang, Ling. / Recent progress and challenges in screening and characterization of UGT1A1 inhibitors. Julkaisussa: Acta pharmaceutica sinica b. 2019 ; Vuosikerta 9, Nro 2. Sivut 258-278.
@article{f4720175c2a24966996eafdaa45a4d0c,
title = "Recent progress and challenges in screening and characterization of UGT1A1 inhibitors",
keywords = "UGT1A1 inhibitors, Drug/herbdrug interactions, Probe substrates, High-throughput screening, UDP-GLUCURONOSYLTRANSFERASE 1A1, HUMAN LIVER-MICROSOMES, RATIOMETRIC FLUORESCENT-PROBE, PRIMARY HUMAN HEPATOCYTES, HUMAN CARBOXYLESTERASE 2, IN-VITRO INHIBITION, BILIRUBIN GLUCURONIDATION, GENETIC-POLYMORPHISM, DRUG-INTERACTIONS, ENZYME-ACTIVITIES, 116 Chemical sciences, 317 Pharmacy",
author = "Xia Lv and Yangliu Xia and Moshe Finel and Jingjing Wu and Guangbo Ge and Ling Yang",
year = "2019",
month = "3",
doi = "10.1016/j.apsb.2018.09.005",
language = "English",
volume = "9",
pages = "258--278",
journal = "Acta pharmaceutica sinica b",
issn = "2211-3835",
publisher = "Elsevier",
number = "2",

}

Recent progress and challenges in screening and characterization of UGT1A1 inhibitors. / Lv, Xia; Xia, Yangliu; Finel, Moshe; Wu, Jingjing; Ge, Guangbo; Yang, Ling.

julkaisussa: Acta pharmaceutica sinica b, Vuosikerta 9, Nro 2, 03.2019, s. 258-278.

Tutkimustuotos: ArtikkelijulkaisuKatsausartikkeliTieteellinenvertaisarvioitu

TY - JOUR

T1 - Recent progress and challenges in screening and characterization of UGT1A1 inhibitors

AU - Lv, Xia

AU - Xia, Yangliu

AU - Finel, Moshe

AU - Wu, Jingjing

AU - Ge, Guangbo

AU - Yang, Ling

PY - 2019/3

Y1 - 2019/3

KW - UGT1A1 inhibitors

KW - Drug/herbdrug interactions

KW - Probe substrates

KW - High-throughput screening

KW - UDP-GLUCURONOSYLTRANSFERASE 1A1

KW - HUMAN LIVER-MICROSOMES

KW - RATIOMETRIC FLUORESCENT-PROBE

KW - PRIMARY HUMAN HEPATOCYTES

KW - HUMAN CARBOXYLESTERASE 2

KW - IN-VITRO INHIBITION

KW - BILIRUBIN GLUCURONIDATION

KW - GENETIC-POLYMORPHISM

KW - DRUG-INTERACTIONS

KW - ENZYME-ACTIVITIES

KW - 116 Chemical sciences

KW - 317 Pharmacy

U2 - 10.1016/j.apsb.2018.09.005

DO - 10.1016/j.apsb.2018.09.005

M3 - Review Article

VL - 9

SP - 258

EP - 278

JO - Acta pharmaceutica sinica b

JF - Acta pharmaceutica sinica b

SN - 2211-3835

IS - 2

ER -