Preparation of N-​fluoropyrrolidin-​2-​ylmethoxy-​7-​oxo-​6-​(sulfooxy)​-​1,​6-​diazabicyclo[3.2.1]​octane-​2-​carboxamide derivatives as antibacterial compounds.

Piyush Patel, Vijaykumar Jagdishwar Patil, Ravikumar Tadiparthi, Rajib Bhuniya, Sachin Bhagwat, Swapna Shripad Takalkar, Rajesh Chavan, Anusuya Patel, Vipul Rane, Mahesh Vithalbhai. Patel

Forskningsoutput: PatentVetenskaplig

Sammanfattning

Disclosed are compds. of formula I, their prepn., and use in preventing or treating a bacterial infection. Compds. of I [wherein R1 - R3 are independently H, CN, halo, aryl, etc.; n = 0, 1, 2, 3 or 4; M = H or cation] and stereoisomers, pharmaceutically acceptable salt thereof, are claimed and exemplified. Example compd. II was prepd. by a multistep procedure (prepn. given). Candidate compds. of I were evaluated for their antibacterial activity (data given). [on SciFinder(R)]
Originalspråkengelska
Utgivningsår21 dec 2017
StatusPublicerad - 21 dec 2017
MoE-publikationstypH1 Beviljat patent

Bibliografisk information

M1 - Copyright (C) 2019 American Chemical Society (ACS). All Rights Reserved.

CAPLUS AN 2017:2002960(Patent)

Citera det här

Patel, P., Patil, V. J., Tadiparthi, R., Bhuniya, R., Bhagwat, S., Takalkar, S. S., ... Patel, M. V. (2017). Preparation of N-​fluoropyrrolidin-​2-​ylmethoxy-​7-​oxo-​6-​(sulfooxy)​-​1,​6-​diazabicyclo[3.2.1]​octane-​2-​carboxamide derivatives as antibacterial compounds. (Patentnr. WO2018158619A1). PCT Int. Appl.
Patel, Piyush (Författare) ; Patil, Vijaykumar Jagdishwar (Författare) ; Tadiparthi, Ravikumar (Författare) ; Bhuniya, Rajib (Författare) ; Bhagwat, Sachin (Författare) ; Takalkar, Swapna Shripad (Författare) ; Chavan, Rajesh (Författare) ; Patel, Anusuya (Författare) ; Rane, Vipul (Författare) ; Patel, Mahesh Vithalbhai. (Författare). / Preparation of N-​fluoropyrrolidin-​2-​ylmethoxy-​7-​oxo-​6-​(sulfooxy)​-​1,​6-​diazabicyclo[3.2.1]​octane-​2-​carboxamide derivatives as antibacterial compounds. PCT Int. Appl. Patentnr.: WO2018158619A1.
@misc{0cdea29672b04617b01ba7460d32c79e,
title = "Preparation of N-​fluoropyrrolidin-​2-​ylmethoxy-​7-​oxo-​6-​(sulfooxy)​-​1,​6-​diazabicyclo[3.2.1]​octane-​2-​carboxamide derivatives as antibacterial compounds.",
abstract = "Disclosed are compds. of formula I, their prepn., and use in preventing or treating a bacterial infection. Compds. of I [wherein R1 - R3 are independently H, CN, halo, aryl, etc.; n = 0, 1, 2, 3 or 4; M = H or cation] and stereoisomers, pharmaceutically acceptable salt thereof, are claimed and exemplified. Example compd. II was prepd. by a multistep procedure (prepn. given). Candidate compds. of I were evaluated for their antibacterial activity (data given). [on SciFinder(R)]",
author = "Piyush Patel and Patil, {Vijaykumar Jagdishwar} and Ravikumar Tadiparthi and Rajib Bhuniya and Sachin Bhagwat and Takalkar, {Swapna Shripad} and Rajesh Chavan and Anusuya Patel and Vipul Rane and Patel, {Mahesh Vithalbhai.}",
note = "M1 - Copyright (C) 2019 American Chemical Society (ACS). All Rights Reserved. CAPLUS AN 2017:2002960(Patent); WO2018158619A1",
year = "2017",
month = "12",
day = "21",
language = "English",
publisher = "PCT Int. Appl",
address = "United States",
type = "Patent",

}

Patel, P, Patil, VJ, Tadiparthi, R, Bhuniya, R, Bhagwat, S, Takalkar, SS, Chavan, R, Patel, A, Rane, V & Patel, MV 2017, Preparation of N-​fluoropyrrolidin-​2-​ylmethoxy-​7-​oxo-​6-​(sulfooxy)​-​1,​6-​diazabicyclo[3.2.1]​octane-​2-​carboxamide derivatives as antibacterial compounds., Patentnr. WO2018158619A1.

Preparation of N-​fluoropyrrolidin-​2-​ylmethoxy-​7-​oxo-​6-​(sulfooxy)​-​1,​6-​diazabicyclo[3.2.1]​octane-​2-​carboxamide derivatives as antibacterial compounds. / Patel, Piyush; Patil, Vijaykumar Jagdishwar; Tadiparthi, Ravikumar; Bhuniya, Rajib; Bhagwat, Sachin; Takalkar, Swapna Shripad; Chavan, Rajesh; Patel, Anusuya; Rane, Vipul; Patel, Mahesh Vithalbhai.

PCT Int. Appl. Patentnr.: WO2018158619A1.

Forskningsoutput: PatentVetenskaplig

TY - PAT

T1 - Preparation of N-​fluoropyrrolidin-​2-​ylmethoxy-​7-​oxo-​6-​(sulfooxy)​-​1,​6-​diazabicyclo[3.2.1]​octane-​2-​carboxamide derivatives as antibacterial compounds.

AU - Patel, Piyush

AU - Patil, Vijaykumar Jagdishwar

AU - Tadiparthi, Ravikumar

AU - Bhuniya, Rajib

AU - Bhagwat, Sachin

AU - Takalkar, Swapna Shripad

AU - Chavan, Rajesh

AU - Patel, Anusuya

AU - Rane, Vipul

AU - Patel, Mahesh Vithalbhai.

N1 - M1 - Copyright (C) 2019 American Chemical Society (ACS). All Rights Reserved. CAPLUS AN 2017:2002960(Patent)

PY - 2017/12/21

Y1 - 2017/12/21

N2 - Disclosed are compds. of formula I, their prepn., and use in preventing or treating a bacterial infection. Compds. of I [wherein R1 - R3 are independently H, CN, halo, aryl, etc.; n = 0, 1, 2, 3 or 4; M = H or cation] and stereoisomers, pharmaceutically acceptable salt thereof, are claimed and exemplified. Example compd. II was prepd. by a multistep procedure (prepn. given). Candidate compds. of I were evaluated for their antibacterial activity (data given). [on SciFinder(R)]

AB - Disclosed are compds. of formula I, their prepn., and use in preventing or treating a bacterial infection. Compds. of I [wherein R1 - R3 are independently H, CN, halo, aryl, etc.; n = 0, 1, 2, 3 or 4; M = H or cation] and stereoisomers, pharmaceutically acceptable salt thereof, are claimed and exemplified. Example compd. II was prepd. by a multistep procedure (prepn. given). Candidate compds. of I were evaluated for their antibacterial activity (data given). [on SciFinder(R)]

M3 - Patent

M1 - WO2018158619A1

PB - PCT Int. Appl

ER -