Recent progress and challenges in screening and characterization of UGT1A1 inhibitors

Xia Lv, Yangliu Xia, Moshe Finel, Jingjing Wu, Guangbo Ge, Ling Yang

Forskningsoutput: TidskriftsbidragÖversiktsartikelVetenskapligPeer review

Originalspråkengelska
TidskriftActa pharmaceutica sinica b
Volym9
Utgåva2
Sidor (från-till)258-278
Antal sidor21
ISSN2211-3835
DOI
StatusPublicerad - mar 2019
MoE-publikationstypA2 Granska artikel i en vetenskaplig tidskrift

Vetenskapsgrenar

  • 116 Kemi
  • 317 Farmaci

Citera det här

Lv, Xia ; Xia, Yangliu ; Finel, Moshe ; Wu, Jingjing ; Ge, Guangbo ; Yang, Ling. / Recent progress and challenges in screening and characterization of UGT1A1 inhibitors. I: Acta pharmaceutica sinica b. 2019 ; Vol. 9, Nr. 2. s. 258-278.
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title = "Recent progress and challenges in screening and characterization of UGT1A1 inhibitors",
keywords = "UGT1A1 inhibitors, Drug/herbdrug interactions, Probe substrates, High-throughput screening, UDP-GLUCURONOSYLTRANSFERASE 1A1, HUMAN LIVER-MICROSOMES, RATIOMETRIC FLUORESCENT-PROBE, PRIMARY HUMAN HEPATOCYTES, HUMAN CARBOXYLESTERASE 2, IN-VITRO INHIBITION, BILIRUBIN GLUCURONIDATION, GENETIC-POLYMORPHISM, DRUG-INTERACTIONS, ENZYME-ACTIVITIES, 116 Chemical sciences, 317 Pharmacy",
author = "Xia Lv and Yangliu Xia and Moshe Finel and Jingjing Wu and Guangbo Ge and Ling Yang",
year = "2019",
month = "3",
doi = "10.1016/j.apsb.2018.09.005",
language = "English",
volume = "9",
pages = "258--278",
journal = "Acta pharmaceutica sinica b",
issn = "2211-3835",
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Recent progress and challenges in screening and characterization of UGT1A1 inhibitors. / Lv, Xia; Xia, Yangliu; Finel, Moshe; Wu, Jingjing; Ge, Guangbo; Yang, Ling.

I: Acta pharmaceutica sinica b, Vol. 9, Nr. 2, 03.2019, s. 258-278.

Forskningsoutput: TidskriftsbidragÖversiktsartikelVetenskapligPeer review

TY - JOUR

T1 - Recent progress and challenges in screening and characterization of UGT1A1 inhibitors

AU - Lv, Xia

AU - Xia, Yangliu

AU - Finel, Moshe

AU - Wu, Jingjing

AU - Ge, Guangbo

AU - Yang, Ling

PY - 2019/3

Y1 - 2019/3

KW - UGT1A1 inhibitors

KW - Drug/herbdrug interactions

KW - Probe substrates

KW - High-throughput screening

KW - UDP-GLUCURONOSYLTRANSFERASE 1A1

KW - HUMAN LIVER-MICROSOMES

KW - RATIOMETRIC FLUORESCENT-PROBE

KW - PRIMARY HUMAN HEPATOCYTES

KW - HUMAN CARBOXYLESTERASE 2

KW - IN-VITRO INHIBITION

KW - BILIRUBIN GLUCURONIDATION

KW - GENETIC-POLYMORPHISM

KW - DRUG-INTERACTIONS

KW - ENZYME-ACTIVITIES

KW - 116 Chemical sciences

KW - 317 Pharmacy

U2 - 10.1016/j.apsb.2018.09.005

DO - 10.1016/j.apsb.2018.09.005

M3 - Review Article

VL - 9

SP - 258

EP - 278

JO - Acta pharmaceutica sinica b

JF - Acta pharmaceutica sinica b

SN - 2211-3835

IS - 2

ER -